SCHEMBL24528629

SCHEMBL24528629

O=Cc1ccc(-c2nc(-c3ccc(C=O)cc3)c3ccsc3n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.45
GGPS1 O95749 5/20 0.39
FDPS P14324 1/20 0.39
PTGS1 P23219 1/20 0.38
CYP2A6 P11509 1/20 0.37
PDE4B Q07343 1/20 0.36
CHEK1 O14757 1/20 0.34
AURKA O14965 1/20 0.34
DAPK3 O43293 1/20 0.34
JAK2 O60674 1/20 0.34
ABL1 P00519 1/20 0.34
NTRK1 P04629 1/20 0.34
CSF1R P07333 1/20 0.34
RET P07949 1/20 0.34
IGF1R P08069 1/20 0.34
PDGFRB P09619 1/20 0.34
PIM1 P11309 1/20 0.34
FGFR1 P11362 1/20 0.34
PRKACA P17612 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29681221 1.00 ADORA2A (0.45) ADORA2AGGPS1FDPSPTGS1CYP2A6
SCHEMBL29680643 0.83 PTGS1 (0.37) ADORA2APTGS1CYP2A6CHEK1AURKA
SCHEMBL24528684 0.83 PTGS1 (0.37) ADORA2APTGS1CYP2A6CHEK1AURKA
SCHEMBL16685612 0.80 ADORA2A (0.68) ADORA2AGGPS1FDPSPDE4BDHODH
SCHEMBL29681010 0.77 MTOR (0.39) ADORA2APTGS1CYP2A6PDE4BMAPT
SCHEMBL24528637 0.77 MTOR (0.39) ADORA2APTGS1CYP2A6PDE4BMAPT
SCHEMBL23637787 0.73 ALDH1A1 (0.46) CYP2A6ALDH1A1MAPT
SCHEMBL24528664 0.73 ADORA2A (0.34) ADORA2AALDH1A1LMNA
SCHEMBL30488661 0.71 DRD1 (0.45) CYP2A6ALDH1A1MAPT
SCHEMBL19106711 0.69 ADORA2A (0.49) ADORA2AAURKAAURKBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed