SCHEMBL24528660

SCHEMBL24528660

CN1CCN(CCC/N=C\c2ccc(-c3nc(-c4ccc(/C=N/CCCN5CCN(C)CC5)cc4)nc4sccc34)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX15 P16050 1/20 0.34
ADORA2A P29274 1/20 0.34
ENPP2 Q13822 1/20 0.33
CXCR1 P25024 2/20 0.32
AGER Q15109 2/20 0.32
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PRKCI P41743 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
TLR9 Q9NR96 2/20 0.31
RAD52 P43351 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29681239 1.00 KDM4E (0.40) KDM4EALDH1A1ALOX15ADORA2AENPP2
SCHEMBL24528662 0.90 ALDH1A1 (0.36) KDM4EALDH1A1ALOX15ADORA2ASMN1; SMN2
SCHEMBL29681009 0.85 KDM4E (0.40) KDM4EALDH1A1ALOX15CXCR1NPC1
SCHEMBL24528587 0.85 KDM4E (0.40) KDM4EALDH1A1ALOX15CXCR1NPC1
SCHEMBL24528685 0.82 KDM4E (0.40) KDM4EALDH1A1ALOX15CXCR1AGER
SCHEMBL29681200 0.82 KDM4E (0.40) KDM4EALDH1A1ALOX15CXCR1AGER
SCHEMBL24528664 0.81 ADORA2A (0.34) KDM4EALDH1A1ADORA2A
SCHEMBL29680554 0.78 RAD52 (0.37) KDM4EALDH1A1NPC1MAPTMAPK1
SCHEMBL24528648 0.78 RAD52 (0.37) KDM4EALDH1A1NPC1MAPTMAPK1
SCHEMBL29680577 0.77 AKT1 (0.47) KDM4EALDH1A1ADORA2AHRH3RAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed