SCHEMBL24529017

SCHEMBL24529017

CC1c2ccc(CCC(=O)O)cc2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.44
NR1H3 Q13133 1/20 0.44
GHSR Q92847 13/20 0.43
S1PR1 P21453 1/20 0.42
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528888 0.91 NR1H2 (0.44) NR1H2NR1H3GHSRS1PR1KMT2A
SCHEMBL31680225 0.89 GHSR (0.42) GHSRKMT2ASMN1; SMN2
SCHEMBL19643138 0.89 GHSR (0.42) GHSRKMT2ASMN1; SMN2
SCHEMBL24529088 0.88 HRH3 (0.41) GHSRKMT2A
SCHEMBL30828033 0.88 HRH3 (0.41) GHSRKMT2A
SCHEMBL18617674 0.86 GHSR (0.43) NR1H2NR1H3GHSRKMT2ASMN1; SMN2
SCHEMBL24528740 0.86 GHSR (0.42) NR1H2GHSRKMT2ASMN1; SMN2
SCHEMBL30828046 0.86 GHSR (0.42) GHSRKMT2A
SCHEMBL24528738 0.86 GHSR (0.42) GHSRKMT2A
SCHEMBL24528998 0.81 NR1H2 (0.43) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263511-A1 NOVEL BIFUNCTIONAL MOLECULES FOR TARGETED PROTEIN DEGRADATION Amphista Therapeutics Ltd (GB) 2023-10-25 EP disclosed
CN-116897150-A Novel bifunctional molecules for protein-targeted degradation 安菲斯塔治疗有限公司 2023-10-17 CN disclosed
WO-2022129925-A1 NOVEL BIFUNCTIONAL MOLECULES FOR TARGETED PROTEIN DEGRADATION AMPHISTA THERAPEUTICS LIMITED (GB) 2022-06-23 WO disclosed
WO-2022129925-A1 NOVEL BIFUNCTIONAL MOLECULES FOR TARGETED PROTEIN DEGRADATION AMPHISTA THERAPEUTICS LIMITED (GB) 2022-06-23 WO disclosed