SCHEMBL24533974

SCHEMBL24533974

CN1CCN(Cc2ncc(N=C(c3ccccc3)c3ccccc3)cc2C(F)(F)F)CC1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RET P07949 10/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
NR1H2 P55055 1/20 0.40
PDGFRB P09619 2/20 0.40
KDR P35968 2/20 0.40
BRAF P15056 3/20 0.39
EGFR P00533 2/20 0.38
MC4R P32245 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21632663 0.78 MC4R (0.43) PDGFRBKDRMC4R
SCHEMBL21465752 0.73 NR1H2 (0.59) RETKDM4EALDH1A1POLBNR1H2
SCHEMBL24533977 0.73 NR1H2 (0.46) RETKDM4EALDH1A1POLBNR1H2
SCHEMBL21465801 0.71 KIT (0.48) BRAFEGFR
SCHEMBL21470482 0.71 GAA (0.48) RETBRAFEGFR
SCHEMBL24191972 0.70 DDR1 (0.44) KDM4EALDH1A1POLBNR1H2PDGFRB
SCHEMBL20483488 0.69 KDM4E (0.38) KDM4EALDH1A1POLBPDGFRBKDR
SCHEMBL30486114 0.68 EGFR (0.46) RETBRAFEGFR
SCHEMBL25220250 0.68 TSHR (0.39) ALDH1A1NR1H2PDGFRBKDRMEN1
SCHEMBL21470484 0.68 FGFR4 (0.41) RETKDM4EALDH1A1POLBNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022128850-A1 NOVEL ISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2022-06-23 WO disclosed