SCHEMBL24533977

SCHEMBL24533977

CN1CCN(Cc2ncc(Br)cc2C(F)(F)F)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.46
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 4/20 0.43
POLB P06746 1/20 0.43
SSTR4 P31391 1/20 0.43
MAPT P10636 2/20 0.38
CHKA P35790 1/20 0.36
GAA P10253 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTR6 P50406 1/20 0.35
CTSS P25774 2/20 0.35
CTSK P43235 2/20 0.35
SRC P12931 1/20 0.35
KCNH2 Q12809 1/20 0.35
MAOB P27338 1/20 0.35
EGFR P00533 2/20 0.35
BRAF P15056 2/20 0.35
FGFR4 P22455 1/20 0.35
RET P07949 1/20 0.34
PTK2 Q05397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21465752 0.83 NR1H2 (0.59) NR1H2ALDH1A1KDM4EPOLBMAPT
SCHEMBL20160565 0.81 TNKS (0.41) ALDH1A1KDM4EMAPTCHKAGAA
SCHEMBL21470484 0.77 FGFR4 (0.41) NR1H2ALDH1A1KDM4EPOLBSRC
SCHEMBL21465801 0.76 KIT (0.48) SRCEGFRBRAFFGFR4
SCHEMBL30486114 0.75 EGFR (0.46) SRCEGFRBRAFFGFR4RET
SCHEMBL24533974 0.73 RET (0.43) NR1H2ALDH1A1KDM4EPOLBEGFR
SCHEMBL21551702 0.71 KDM4E (0.45) ALDH1A1KDM4EMAPTCHKAGAA
SCHEMBL2067677 0.71 HTT (0.35) SSTR4
SCHEMBL1577283 0.71 CYP11B1 (0.35) SSTR4
SCHEMBL1252213 0.70 GAA (0.48) NR1H2ALDH1A1KDM4EPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022128850-A1 NOVEL ISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2022-06-23 WO disclosed