SCHEMBL2454259

SCHEMBL2454259

NC1CCC2CN(S(=O)(=O)c3ccc(C(F)(F)F)cc3Cl)CC12

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 13/20 0.47
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CACNA1B Q00975 3/20 0.42
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65327 1.00 TRPV4 (0.47) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL2454255 1.00 TRPV4 (0.47) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL2458246 1.00 TRPV4 (0.47) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL2420763 0.86 TRPV4 (0.47) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL65565 0.83 CACNA1B (0.49) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL67623 0.81 CACNA1B (0.50) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL67995 0.81 CACNA1B (0.49) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL65932 0.81 TRPV4 (0.45) TRPV4MEN1ALDH1A1TSHRKMT2A
SCHEMBL2419370 0.80 CACNA1B (0.57) MEN1ALDH1A1KMT2AL3MBTL1CACNA1B
SCHEMBL16497951 0.80 CACNA1B (0.57) MEN1ALDH1A1KMT2AL3MBTL1CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149995-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA [C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2011-12-01 WO disclosed
EP-2367790-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS Abbott Laboratories (US) 2011-09-28 EP disclosed