SCHEMBL245487

SCHEMBL245487

C#Cc1cccc(Nc2ncnc3cc(OC)c(N(C)C(=O)N4C[C@H]5CCN[C@H]5C4)cc23)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.56
GAK O14976 3/20 0.55
FBP1 P09467 2/20 0.55
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
HDAC3 O15379 7/20 0.51
HDAC4 P56524 7/20 0.51
HDAC1 Q13547 7/20 0.51
HDAC7 Q8WUI4 7/20 0.51
HDAC2 Q92769 7/20 0.51
HDAC10 Q969S8 7/20 0.51
HDAC11 Q96DB2 7/20 0.51
HDAC8 Q9BY41 7/20 0.51
HDAC6 Q9UBN7 7/20 0.51
HDAC9 Q9UKV0 7/20 0.51
HDAC5 Q9UQL6 7/20 0.51
ERBB2 P04626 7/20 0.50
RIPK2 O43353 2/20 0.49
BUB1 O43683 2/20 0.49
STK10 O94804 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13514680 0.75 EGFR (0.66) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL13514684 0.74 EGFR (0.64) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL13514688 0.74 EGFR (0.67) EGFRGAKFBP1ALDH1A1MAPT
Theliatinib SCHEMBL29370993 0.73 EGFR (0.62) EGFRGAKFBP1ALDH1A1MAPT
Theliatinib SCHEMBL247509 0.73 EGFR (0.62) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL667895 0.73 EGFR (1.00) EGFRGAKFBP1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL1507455 0.72 EGFR (0.98) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL14489912 0.72 EGFR (0.72) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL29623598 0.72 EGFR (0.69) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL185131 0.72 EGFR (0.69) EGFRGAKFBP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590966-A1 QUINAZOLINE COMPOUNDS Hutchison Medipharma Limited (CN) 2013-05-15 EP disclosed
WO-2012000356-A1 QUINAZOLINE COMPOUNDS HUTCHISON MEDIPHARMA LIMITED (CN) 2012-01-05 WO disclosed