SCHEMBL29623598

SCHEMBL29623598

C#Cc1cccc(Nc2ncnc3cc(OC)c(OC4CCN(C(C)=O)CC4)cc23)c1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.69
GAK O14976 1/20 0.68
ALDH1A1 P00352 1/20 0.68
FBP1 P09467 1/20 0.68
MAPT P10636 1/20 0.68
ERBB2 P04626 5/20 0.65
HDAC3 O15379 2/20 0.60
HDAC4 P56524 2/20 0.60
HDAC1 Q13547 2/20 0.60
HDAC7 Q8WUI4 2/20 0.60
HDAC2 Q92769 2/20 0.60
HDAC10 Q969S8 2/20 0.60
HDAC11 Q96DB2 2/20 0.60
HDAC8 Q9BY41 2/20 0.60
HDAC6 Q9UBN7 2/20 0.60
HDAC9 Q9UKV0 2/20 0.60
HDAC5 Q9UQL6 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL185131 1.00 EGFR (0.69) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL14489912 0.94 EGFR (0.72) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL3433430 0.91 EGFR (0.83) EGFRERBB2
SCHEMBL1943518 0.91 EGFR (0.69) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL12754569 0.91 EGFR (0.67) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL12536553 0.91 EGFR (0.66) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL12536562 0.91 EGFR (0.66) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL14489872 0.91 EGFR (0.66) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL14489910 0.91 EGFR (0.66) EGFRGAKALDH1A1FBP1MAPT
SCHEMBL226341 0.91 EGFR (0.66) EGFRGAKALDH1A1FBP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110840847-B Pharmaceutical compositions for the treatment of cystic fibrosis transmembrane conductance regulator mediated diseases 沃泰克斯药物股份有限公司 2022-07-29 CN disclosed
CN-110713489-B Heteroaryl SYK inhibitors 勃林格殷格翰国际有限公司 2022-05-31 CN disclosed
CN-110183440-B Heteroaryl SYK inhibitors 勃林格殷格翰国际有限公司 2022-04-22 CN disclosed