SCHEMBL2456643

SCHEMBL2456643

C#CCO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
BLM P54132 1/20 0.36
CYP3A4 P08684 2/20 0.34
HTT P42858 1/20 0.34
MAOB P27338 6/20 0.33
MAOA P21397 3/20 0.33
PYCR1 P32322 2/20 0.33
NPC1 O15118 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
KCNH3 Q9ULD8 1/20 0.33
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2188878 0.83 SMYD2 (0.37) SMYD2SMN1; SMN2LMNAALDH1A1BLM
SCHEMBL17496700 0.83 SMYD2 (0.33) SMYD2SMN1; SMN2LMNAALDH1A1BLM
SCHEMBL3638318 0.81 SMYD2 (0.36) SMYD2SMN1; SMN2CYP3A4HTT
SCHEMBL3456559 0.80 SMYD2 (0.36) SMYD2SMN1; SMN2CYP3A4HTT
SCHEMBL31092036 0.79 SMYD2 (0.37) SMYD2SMN1; SMN2ALDH1A1CYP3A4HTT
SCHEMBL9468934 0.79 CYP3A4 (0.33) SMYD2SMN1; SMN2CYP3A4HTT
SCHEMBL3262971 0.79 CYP3A4 (0.35) SMYD2SMN1; SMN2ALDH1A1CYP3A4HTT
SCHEMBL6795155 0.79 CYP3A4 (0.35) SMYD2SMN1; SMN2CYP3A4HTT
SCHEMBL9468930 0.79 CYP3A4 (0.33) SMYD2SMN1; SMN2CYP3A4HTT
SCHEMBL17093480 0.78 SMYD2 (0.34) SMYD2SMN1; SMN2CYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624044-B2 SMARCA degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2026-05-12 US disclosed
WO-2025124516-A1 COMPOUND HAVING AKT KINASE-DEGRADING ACTIVITY, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 南京正大天晴制药有限公司 2025-06-19 WO disclosed
CN-120157686-A Compound with AKT kinase degradation activity, preparation method and pharmaceutical application thereof 南京正大天晴制药有限公司 2025-06-17 CN disclosed
CN-118994171-A Preparation method of rebamacinib intermediate 2-chloro-7-cyclopentyl-7H-pyrrolo [2,3-d ] pyrimidine-6-methanol 浙江工业大学 2024-11-22 CN disclosed
US-20230381189-A1 TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY G1 THERAPEUTICS, INC. (US) 2023-11-30 US disclosed
US-20230364098-A1 HSPC-SPARING TREATMENTS FOR RB-POSITIVE ABNORMAL CELLULAR PROLIFERATION G1 THERAPEUTICS, INC. (US) 2023-11-16 US disclosed
US-20230248733-A1 HIGHLY ACTIVE ANTI-NEOPLASTIC AND ANTI-PROLIFERATIVE AGENTS G1 THERAPEUTICS, INC. (US) 2023-08-10 US disclosed
US-11717523-B2 Transient protection of normal cells during chemotherapy G1 THERAPEUTICS, INC. (US) 2023-08-08 US disclosed
US-20230241059-A1 ANTI-NEOPLASTIC COMBINATIONS AND DOSING REGIMENS USING CDK4/6 INHIBITOR COMPOUNDS TO TREAT RB-POSITIVE TUMORS G1 THERAPEUTICS, INC. (US) 2023-08-03 US disclosed
US-11654148-B2 HSPC-sparing treatments for RB-positive abnormal cellular proliferation G1 THERAPEUTICS, INC. (US) 2023-05-23 US disclosed
WO-2011106997-A1 NOVEL 10-23 DEOXYRIBOZYME ANALOGUES AND USES THEREOF 中国人民解放军军事医学科学院毒物药物研究所 (CN) 2011-09-09 WO disclosed
WO-2007134421-A1 2-VINYL INDOLES, PYRIDO AND AZEPINO INDOLE DERIVATIVES, 2-ALKYNYL INDOLES, 2-ALKYNYL BENZO[b]FURANS, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2007-11-29 WO disclosed
US-5527805-A DNA-CLEAVING, CYTOTOXIC AND ANTI-TUMOR COMPOUNDS THE SCRIPPS RESEARCH INSTITUTE (US) 1996-06-18 US disclosed
EP-0523151-B1 TRANSMETALATIONS FROM ZIRCONIUM TO COPPER INTERMEDIATES UNIV CALIFORNIA (US) 1994-12-28 EP disclosed
US-5286889-A Reacting 1-alkyne with zirconocene chloride hydride, reacting product with organic lithium compound, reacting with lithium cuprate compound REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-02-15 US disclosed
US-5281710-A Antibiotics or antitumor agents THE SCRIPPS RESEARCH INSTITUTE (US) 1994-01-25 US disclosed
US-5276159-A Antitumor THE SCRIPPS RESEARCH INSTITUTE (US) 1994-01-04 US disclosed
US-5072010-A Reacting zirconium and lithium compounds, reacting product with copper/lithium complex UNIVERSITY OF CALIFORNIA (US) 1991-12-10 US disclosed
US-4959391-A LIPOXYGENASE INHIBITORS, LEUKOTRIENE DISEASES GRUENENTHAL GMBH (DE) 1990-09-25 US disclosed
US-4760087-A 5-lipoxygenase inhibitor GRUENENTHAL GMBH (DE) 1988-07-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230364098-A1 HSPC-SPARING TREATMENTS FOR RB-POSITIVE ABNORMAL CELLULAR PROLIFERATION RB1, CDK4, CDKN1A SMYD2 623/4885SMN1; SMN2 751/4885LMNA 2987/4885
US-20230248733-A1 HIGHLY ACTIVE ANTI-NEOPLASTIC AND ANTI-PROLIFERATIVE AGENTS MKI67, PCNA, HRAS SMYD2 1157/4885SMN1; SMN2 2179/4885LMNA 1553/4885
US-20230381189-A1 TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY CDK6, CCNC, MCL1 SMYD2 2274/4885SMN1; SMN2 2529/4885LMNA 2729/4885
US-12624044-B2 SMARCA degraders and uses thereof SMARCA1, SMARCC1, SMARCA2 SMYD2 569/4885SMN1; SMN2 326/4885LMNA 746/4885
US-20230241059-A1 ANTI-NEOPLASTIC COMBINATIONS AND DOSING REGIMENS USING CDK4/6 INHIBITOR COMPOUNDS TO TREAT RB-POSITIVE TUMORS CDK4, RB1, BTK SMYD2 1950/4885SMN1; SMN2 2678/4885LMNA 2259/4885
US-11654148-B2 HSPC-sparing treatments for RB-positive abnormal cellular proliferation RB1, CDK4, CDKN1A SMYD2 623/4885SMN1; SMN2 751/4885LMNA 2987/4885
US-11717523-B2 Transient protection of normal cells during chemotherapy CDK6, CCNC, MCL1 SMYD2 2274/4885SMN1; SMN2 2529/4885LMNA 2729/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.