SCHEMBL24575288

SCHEMBL24575288

O=C(C1CCOCC1)N1CC2C[C@@H](Nc3nnc(Cl)cc3C3CC3)C[C@@H]2C1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATXN2 Q99700 2/20 0.45
JAK1 P23458 6/20 0.42
AURKA O14965 4/20 0.42
PIK3CD O00329 4/20 0.35
PIK3CA P42336 2/20 0.35
PIK3R1 P27986 2/20 0.35
EPHX2 P34913 3/20 0.34
GRM5 P41594 1/20 0.34
CNR2 P34972 3/20 0.33
AURKB Q96GD4 2/20 0.33
JAK2 O60674 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
FLT3 P36888 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31119103 1.00 ATXN2 (0.45) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL23499431 0.88 JAK1 (0.40) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL23499428 0.88 JAK1 (0.40) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL23499430 0.88 JAK1 (0.40) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL23499425 0.84 JAK1 (0.42) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL23499427 0.84 JAK1 (0.42) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL29919210 0.84 AURKA (0.42) JAK1AURKAPIK3CDPIK3CAPIK3R1
SCHEMBL23933530 0.84 JAK1 (0.41) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL23933533 0.84 JAK1 (0.41) ATXN2JAK1AURKAPIK3CDPIK3CA
SCHEMBL23499423 0.84 JAK1 (0.36) ATXN2JAK1AURKAAURKBJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023102100-A1 ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2023-06-08 WO disclosed
WO-2022140499-A1 ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2022-06-30 WO disclosed