Tetrahydrocannabivarin

Tetrahydrocannabivarin

SCHEMBL245827

CCCc1cc(O)c2c(c1)OC(C)(C)C1CCC(C)=CC21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 16/20 1.00
CNR1 P21554 14/20 1.00
TRPM8 Q7Z2W7 2/20 1.00
GPR55 Q9Y2T6 2/20 1.00
TRPA1 O75762 1/20 1.00
HTR1A P08908 1/20 1.00
TRPV1 Q8NER1 1/20 1.00
TRPV3 Q8NET8 1/20 1.00
TRPV6 Q9H1D0 1/20 1.00
TRPV4 Q9HBA0 1/20 1.00
TRPV5 Q9NQA5 1/20 1.00
TRPV2 Q9Y5S1 1/20 1.00
ABHD12 Q8N2K0 3/20 0.86
ABHD6 Q9BV23 3/20 0.86
FAAH O00519 2/20 0.86
NR1I2 O75469 1/20 0.86
LDHA P00338 1/20 0.86
GLRA1 P23415 1/20 0.86
GPR183 P32249 1/20 0.86
DRD3 P35462 1/20 0.86

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tetrahydrocannabivarin SCHEMBL29904669 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL29422123 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL30017852 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL31300003 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL31544930 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL18371743 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL29350511 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL6856739 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL21363566 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1
Tetrahydrocannabivarin SCHEMBL25731794 1.00 CNR2 (1.00) CNR2CNR1TRPM8GPR55TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9593 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4412609-B1 ALKOXYLATION OF CANNABIDIOL & OTHER CANNABINOIDS INDORAMA VENTURES OXIDES LLC (US) 2026-05-27 EP claimed
US-12636251-B1 Glycoside-containing aqueous formulations having a lipophilic active component Doane Technology Group LLC (US) 2026-05-26 US claimed
US-12629332-B2 Cannabinoid chewing gum with sugar alcohols NORDICCAN A/S (DK) 2026-05-19 US claimed
EP-4739284-A1 AN ADHESIVE ORAL DISC FOR SUSTAINED RELEASE OF CANNABINOIDS Fertin Pharma A/S (DK) 2026-05-13 EP claimed
EP-4291170-B1 USE OF CANNABIDIVARIN IN THE TREATMENT OF SEIZURES ASSOCIATED WITH CANINE EPILEPSY JAZZ PHARMACEUTICALS RESEARCH UK LTD (GB) 2026-05-13 EP claimed
EP-4740961-A2 CANNABINOID PRODUCT FOR IMPROVING MUSCULOSKELETAL HEALTH Lonza Greenwood LLC (US) 2026-05-13 EP claimed
EP-4734974-A1 CANNABINOID COMPOSITION FOR USE IN THE TREATMENT OF PAIN AND/OR INFLAMMATION Mabewo Phytopharm AG (CH) 2026-05-06 EP claimed
US-12616728-B2 Processes and systems for converting cannabinoids into cannabinoid derivatives and isolating the same SUPER CRITICAL IP, LLC (US) 2026-05-05 US claimed
EP-4037503-B1 CANNABINOID PRODUCT FOR IMPROVING MUSCULOSKELETAL HEALTH LONZA GREENWOOD LLC (US) 2026-04-29 EP claimed
US-12611446-B2 Cannabinoid product for improving musculoskeletal health LONZA GREENWOOD LLC (US) 2026-04-28 US claimed
US-20110082195-A1 NEW USE FOR CANNABINOIDS GW PHARMA LIMITED (GB) 2011-04-07 US claimed
EP-2283832-A1 Compositions comprising cannabinoids for treatment of nausea, vomiting, emesis, motion sickness or like conditions GW Pharma Limited (GB) 2011-02-16 EP claimed
WO-2011001169-A1 USE OF ONE OR A COMBINATION OF PHYTO-CANNABINOIDS IN THE TREATMENT OF EPILEPSY GW PHARMA LIMITED (GB) 2011-01-06 WO claimed
EP-2161262-A1 THCV and THCV extracts derived from plant material GW Pharma Limited (GB) 2010-03-10 EP claimed
WO-2010013240-A1 COMPOSITIONS AND METHODS FOR TREATING INFLAMMATORY DISORDERS DEKEL PHARMACEUTICALS LTD. (IL) 2010-02-04 WO claimed
US-20070077660-A1 Method for the detection of a cannabinoid, detection kit, and developing solvent GLAS RONALD J 2007-04-05 US claimed
EP-1542984-A2 METHODS OF PURIFYING CANNABINOIDS FROM PLANT MATERIAL GW Pharma Limited (GB) 2005-06-22 EP claimed
WO-2004026857-A2 METHODS OF PURIFYING CANNABINOIDS FROM PLANT MATERIAL GW PHARMA LIMITED (GB) 2004-04-01 WO claimed
EP-1109533-A1 PULMONARY DELIVERY OF LIPOSOME-ENCAPSULATED CANNABINOIDS Hung, Orlando (CA) 2001-06-27 EP claimed
WO-2001003668-A1 PULMONARY DELIVERY OF LIPOSOME-ENCAPSULATED CANNABINOIDS HER MAJESTY THE QUEEN AS REPRESENTED BY THE MINISTER OF NATIONAL DEFENCE OF HER MAJESTY'S CANADIAN GOVERNMENT (CA) 2001-01-18 WO claimed