SCHEMBL24595124

SCHEMBL24595124

CCc1cncc(C#N)c1C(C)C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 12/20 0.40
MAPK1 P28482 1/20 0.34
RIPK1 Q13546 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
CYP2E1 P05181 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2A6 P11509 1/20 0.32
CYP2B6 P20813 1/20 0.32
CYP2C19 P33261 1/20 0.32
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
S1PR1 P21453 1/20 0.30
PARP1 P09874 1/20 0.30
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748960 0.82 KDM5A (0.37) KDM5AKDM5B
SCHEMBL20314862 0.80 SMN1; SMN2 (0.34)
SCHEMBL21937398 0.76 MAPT (0.34) CYP2E1CYP2C8CYP2D6CYP2A6CYP2B6
SCHEMBL21736809 0.76 KDM5A (0.36) KDM5A
SCHEMBL7215529 0.76 KDM5A (0.39) KDM5AMAPK1RIPK1CCNCCDK8
SCHEMBL10058048 0.76 MEN1 (0.38) KDM5AMAPK1RIPK1CCNCCDK8
SCHEMBL21736808 0.74 KDM5A (0.33) KDM5A
SCHEMBL19779742 0.74 CYP2E1 (0.37) KDM5AMAPK1RIPK1CCNCCDK8
SCHEMBL13747989 0.74 CYP11B2 (0.35) KDM5A
SCHEMBL24595067 0.74 KDM5A (0.35) KDM5AKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3636636-B1 PYRIDONE COMPOUND AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE MITSUI CHEMICALS AGRO INC (JP) 2022-07-06 EP disclosed