SCHEMBL24601250

SCHEMBL24601250

CCc1nc(NCc2ccccc2)c2ncn([C@@H]3O[C@H](C(=O)NC)[C@H]4OC(C)(C)O[C@H]43)c2n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 11/20 0.60
ADORA2A P29274 5/20 0.60
ADORA1 P30542 5/20 0.60
ADORA2B P29275 4/20 0.60
MAPK1 P28482 3/20 0.53
MAPT P10636 2/20 0.53
TP53 P04637 2/20 0.53
NPC1 O15118 1/20 0.53
GMNN O75496 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
THRB P10828 1/20 0.53
HPGD P15428 1/20 0.53
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53
KMT2A Q03164 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24600773 0.93 NT5E (0.54) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601008 0.86 ADORA3 (0.57) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601526 0.86 ADORA3 (0.57) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601009 0.86 ADORA3 (0.57) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL29073694 0.86 ADORA3 (0.80) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL29762268 0.86 ADORA3 (0.80) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL29073686 0.86 ADORA3 (0.80) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601270 0.86 ADORA3 (0.80) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24600772 0.85 NT5E (0.56) ADORA3ADORA2AADORA1ADORA2BTP53
SCHEMBL24600730 0.83 ADORA3 (0.58) ADORA3ADORA2AADORA1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4273153-A1 ADENOSINE A3 RECEPTOR AGONISTS, PREPARATION METHODS AND USES THEREOF Zhejiang Vimgreen Pharmaceuticals, Ltd (CN) 2023-11-08 EP disclosed
WO-2022143740-A1 ADENOSINE A3 RECEPTOR AGONIST, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江春禾医药科技有限公司 2022-07-07 WO disclosed