SCHEMBL24601450

SCHEMBL24601450

CCOC(=O)c1cc2cc(NC(=O)c3ccccc3)ccc2[nH]1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 5/20 0.72
MAOA P21397 2/20 0.66
MAOB P27338 2/20 0.66
MMP2 P08253 4/20 0.63
HRH3 Q9Y5N1 1/20 0.62
RAB9A P51151 8/20 0.60
NPC1 O15118 7/20 0.60
SMN1; SMN2 Q16637 5/20 0.60
ALDH1A1 P00352 4/20 0.60
KDM4E B2RXH2 3/20 0.60
HPGD P15428 3/20 0.60
GAA P10253 2/20 0.60
HSD17B10 Q99714 1/20 0.60
LMNA P02545 2/20 0.58
MAPT P10636 2/20 0.58
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
GLA P06280 1/20 0.58
ATM Q13315 1/20 0.58
TP53 P04637 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889575 0.91 MMP13 (0.72) MMP13MAOAMAOBMMP2HRH3
SCHEMBL8204629 0.91 MMP13 (0.76) MMP13MAOAMAOBMMP2HRH3
SCHEMBL8205173 0.88 MMP13 (0.72) MMP13MAOAMAOBMMP2HRH3
SCHEMBL22718539 0.88 MMP13 (0.68) MMP13MAOAMAOBMMP2HRH3
SCHEMBL28941302 0.87 MMP13 (0.58) MMP13MAOAMAOBMMP2HRH3
SCHEMBL28746477 0.87 MMP13 (0.58) MMP13MAOAMAOBMMP2HRH3
SCHEMBL22718574 0.87 MMP13 (0.67) MMP13MAOAMAOBMMP2HRH3
SCHEMBL8204370 0.85 MMP13 (0.83) MMP13MAOAMMP2HRH3RAB9A
SCHEMBL8209912 0.85 MMP13 (0.83) MMP13MAOAMMP2HRH3RAB9A
SCHEMBL22718569 0.84 MMP13 (0.67) MMP13MMP2HRH3RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220213052-A1 INHIBITORS OF RNA-BINDING PROTEINS, COMPOSITIONS THEREOF, AND THERAPEUTIC USES THEROF THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2022-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220213052-A1 INHIBITORS OF RNA-BINDING PROTEINS, COMPOSITIONS THEREOF, AND THERAPEUTIC USES THEROF HNRNPF, RBM3, RBM15 MMP13 3193/4885MAOA 4560/4885MAOB 3990/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.