SCHEMBL24615488

SCHEMBL24615488

CC1(C)OB(c2cc3c(N4CC5CCC(C4)N5C(=O)[C@@H]4C[C@H]4F)ncnn3c2)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 4/20 0.40
JAK1 P23458 4/20 0.40
TYK2 P29597 4/20 0.40
KIT P10721 16/20 0.36
JAK3 P52333 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24615262 0.89 JAK2 (0.40) JAK2JAK1TYK2KITJAK3
SCHEMBL24615465 0.85 TYK2 (0.42) JAK2JAK1TYK2JAK3
SCHEMBL24615451 0.81 JAK2 (0.42) JAK2JAK1TYK2KITJAK3
SCHEMBL24615385 0.79 KIT (0.54) KIT
SCHEMBL24615387 0.79 KIT (0.54) KIT
SCHEMBL24615288 0.79 KIT (0.54) KIT
SCHEMBL24615291 0.79 KIT (0.54) KIT
SCHEMBL24615386 0.77 KIT (0.42) JAK2JAK1TYK2KIT
SCHEMBL24615358 0.76 KIT (0.46) JAK2JAK1TYK2KITJAK3
SCHEMBL24615390 0.76 KIT (0.46) JAK2JAK1TYK2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4274832-A1 TYK2 INHIBITORS Biogen MA Inc. (US) 2023-11-15 EP disclosed
WO-2022150446-A1 TYK2 INHIBITORS BIOGEN MA INC. (US) 2022-07-14 WO disclosed
WO-2022150446-A1 TYK2 INHIBITORS BIOGEN MA INC. (US) 2022-07-14 WO disclosed