SCHEMBL2462437

SCHEMBL2462437

COC(=O)O[C@H]1C[C@@H](O)CN1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.32
CHRNA4 P43681 3/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA7 P36544 1/20 0.32
OGA O60502 1/20 0.32
SMYD3 Q9H7B4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2572486 0.83
SCHEMBL27835327 0.80 CHRM2 (0.33)
Hydrochloric Acid SCHEMBL4427864 0.78 CHRM2 (0.33)
Hydrochloric Acid SCHEMBL27763502 0.78 CHRM2 (0.33)
SCHEMBL1989780 0.78 DPP4 (0.31)
SCHEMBL2562325 0.78 DPP4 (0.31)
SCHEMBL2558329 0.78 DPP4 (0.31)
SCHEMBL5252957 0.76
SCHEMBL5509812 0.76
SCHEMBL9664087 0.75 L3MBTL1 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367815-B1 PYRIDAZINONE DERIVATIVES MERCK PATENT GMBH (DE) 2015-01-14 EP disclosed
EP-2010185-B1 DIHYDROTHIENOPYRIMIDINE FOR TREATING INFLAMMATORY DISORDERS BOEHRINGER INGELHEIM INT (DE) 2012-06-13 EP disclosed
EP-2367815-A1 PYRIDAZINONE DERIVATIVES Merck Patent GmbH (DE) 2011-09-28 EP disclosed
WO-2010072296-A1 PYRIDAZINONE DERIVATIVES MERCK PATENT GMBH (DE) 2010-07-01 WO disclosed
EP-1847543-A1 Dihydrothienopyrimidines for the treatment of inflammatory diseases Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2007-10-24 EP disclosed