SCHEMBL24625529

SCHEMBL24625529

COCCC(NC(=O)OC(C)(C)C)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CTSK P43235 13/20 0.41
CYP2D6 P10635 1/20 0.38
CTSS P25774 4/20 0.38
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
APLNR P35414 1/20 0.36
CA12 O43570 1/20 0.36
CA14 Q9ULX7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24427288 0.83 CA1 (0.44) CA1CA2CA7CTSKCYP2D6
SCHEMBL14533725 0.83 CTSK (0.49) CA1CA2CA7CTSKCTSS
SCHEMBL15425451 0.83 CA1 (0.44) CA1CA2CA7CTSKCYP2D6
SCHEMBL27853976 0.82 CA1 (0.42) CA1CA2CA7CTSKCYP2D6
SCHEMBL16058094 0.82 CA1 (0.38) CA1CA2CA7CTSKCYP2D6
SCHEMBL31059680 0.81 CTSK (0.44) CA1CA2CA7CTSKCYP2D6
SCHEMBL31059691 0.81 TDP1 (0.46) CA1CA2CA7CTSKCYP2D6
SCHEMBL1692753 0.80 CA1 (0.46) CA1CA2CA7CTSKCYP2D6
SCHEMBL31255051 0.80 CA1 (0.46) CA1CA2CA7CTSKCYP2D6
SCHEMBL12330001 0.80 CTSK (0.46) CA1CA2CA7CTSKCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3998260-B1 SGC STIMULATORS CYCLERION THERAPEUTICS INC (US) 2023-11-01 EP disclosed
WO-2022148442-A1 6-SUBSTITUTED PHOSPHORYL QUINAZOLINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-07-14 WO disclosed
WO-2022148442-A1 6-SUBSTITUTED PHOSPHORYL QUINAZOLINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-07-14 WO disclosed
CN-114716478-A 6-substituted phosphoryl quinazoline derivative and preparation method and application thereof 武汉人福创新药物研发中心有限公司 2022-07-08 CN disclosed