SCHEMBL24633865

SCHEMBL24633865

CC(C)(C)OC(=O)[C@H](CCc1ccc(C(F)(F)F)c(F)c1)NC(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 3/20 0.42
TP53 P04637 3/20 0.42
MDM2 Q00987 3/20 0.42
PTPN1 P18031 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29633735 1.00 MDM4 (0.42) MDM4TP53MDM2PTPN1
SCHEMBL28741485 1.00 MDM4 (0.42) MDM4TP53MDM2PTPN1
SCHEMBL24633763 0.91 MDM4 (0.42) MDM4TP53MDM2PTPN1
SCHEMBL29634082 0.91 PTPN1 (0.44) MDM4TP53MDM2PTPN1
SCHEMBL28741600 0.91 MDM4 (0.41) MDM4TP53MDM2PTPN1
SCHEMBL24633884 0.91 MDM4 (0.41) MDM4TP53MDM2PTPN1
SCHEMBL29633743 0.91 MDM4 (0.41) MDM4TP53MDM2PTPN1
SCHEMBL22454533 0.90 MDM4 (0.43) MDM4TP53MDM2PTPN1
SCHEMBL29633764 0.90 MDM4 (0.43) MDM4TP53MDM2PTPN1
SCHEMBL29633746 0.90 MDM4 (0.43) MDM4TP53MDM2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230151060-A1 CYCLIC PEPTIDE COMPOUND HAVING KRAS INHIBITORY ACTION CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-05-18 US disclosed
US-20230151060-A1 CYCLIC PEPTIDE COMPOUND HAVING KRAS INHIBITORY ACTION CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-05-18 US disclosed
WO-2022234853-A1 CYCLIC COMPOUND HAVING INHIBITORY EFFECT SELECTIVE FOR KRAS BUT NOT FOR HRAS AND NRAS 中外製薬株式会社 2022-11-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230151060-A1 CYCLIC PEPTIDE COMPOUND HAVING KRAS INHIBITORY ACTION KRAS, NRAS, HRAS MDM4 441/4885TP53 34/4885MDM2 164/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.