SCHEMBL2463401

SCHEMBL2463401

CC(C)CCNC(=O)Oc1ccc(N2CCN(C(=O)c3ccccc3[N+](=O)[O-])CC2)nn1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCD O00767 4/20 0.52
SMN1; SMN2 Q16637 2/20 0.44
POLB P06746 2/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2468543 0.86 SCD (0.55) SCD
SCHEMBL2468541 0.86 SCD (0.55) SCDALDH1A1
SCHEMBL937950 0.85 SCD (0.71) SCD
SCHEMBL2469229 0.84 SCD (0.74) SCD
SCHEMBL2462941 0.83 SCD (0.52) SCD
SCHEMBL2464963 0.80 SCD (0.49) SCDCYP2C19ALDH1A1HTT
SCHEMBL2464511 0.79 L3MBTL1 (0.56) SCDSMN1; SMN2CYP2C19ALDH1A1
SCHEMBL2464967 0.79 SCD (0.67) SCD
SCHEMBL2466638 0.77 SCD (0.59) SCD
SCHEMBL2464895 0.77 SCD (0.59) SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1648874-B1 PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2011-10-05 EP claimed
EP-1846035-B1 COMBINATION THERAPY XENON PHARMACEUTICALS INC (CA) 2011-09-21 EP claimed