SCHEMBL24639281

SCHEMBL24639281

COc1cnc2c(c1)OCC[C@H]1CN(C(C)C)CCN21

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.38
TIPARP Q7Z3E1 11/20 0.36
PARP2 Q9UGN5 3/20 0.36
KDM2B Q8NHM5 2/20 0.35
HRH3 Q9Y5N1 2/20 0.33
GRM5 P41594 2/20 0.33
ACACB O00763 1/20 0.33
PDE1B Q01064 1/20 0.32
PDE1C Q14123 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24639247 0.89 TIPARP (0.35) TIPARPPARP2KDM2BHRH3GRM5
SCHEMBL24639266 0.89 TIPARP (0.35) TIPARPPARP2KDM2BHRH3GRM5
SCHEMBL24639358 0.85 SOS1 (0.41) SOS1TIPARPPARP2
SCHEMBL24639353 0.85 SOS1 (0.41) SOS1TIPARPPARP2
SCHEMBL24640219 0.84 TIPARP (0.45) SOS1TIPARPPARP2HRH3GRM5
SCHEMBL24639386 0.84 TIPARP (0.45) SOS1TIPARPPARP2HRH3GRM5
SCHEMBL24639388 0.84 TIPARP (0.45) SOS1TIPARPPARP2HRH3GRM5
SCHEMBL24640176 0.83 SOS1 (0.38) SOS1TIPARPPARP2HRH3CYP3A4
SCHEMBL24640221 0.83 SOS1 (0.38) SOS1TIPARPPARP2HRH3CYP3A4
SCHEMBL24640222 0.83 SOS1 (0.38) SOS1TIPARPPARP2HRH3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed