SCHEMBL24639833

SCHEMBL24639833

CC(C)N1CCN2c3ncc(C(F)(F)F)cc3N(CC(F)(F)F)C2C1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.37
NR1H3 Q13133 2/20 0.37
HRH3 Q9Y5N1 4/20 0.36
ACACB O00763 2/20 0.35
CHRM2 P08172 1/20 0.35
HTR1A P08908 1/20 0.35
DRD3 P35462 1/20 0.35
HTR2B P41595 1/20 0.35
MDM2 Q00987 2/20 0.34
TIPARP Q7Z3E1 2/20 0.33
OGA O60502 4/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24639871 0.90 HRH3 (0.37) NR1H2NR1H3HRH3ACACBCHRM2
SCHEMBL24639851 0.84 HRH3 (0.36) NR1H2NR1H3HRH3ACACBCHRM2
SCHEMBL24639861 0.84 HRH3 (0.36) NR1H2NR1H3HRH3ACACBCHRM2
SCHEMBL24640011 0.80 TIPARP (0.40) NR1H2NR1H3HRH3ACACBMDM2
SCHEMBL24640002 0.80 TIPARP (0.40) NR1H2NR1H3HRH3ACACBMDM2
SCHEMBL24639855 0.80 ACACB (0.40) NR1H2NR1H3HRH3ACACBMDM2
SCHEMBL24639836 0.80 HRH3 (0.35) NR1H2NR1H3HRH3ACACBCHRM2
SCHEMBL24639864 0.79 HRH3 (0.33) NR1H2NR1H3HRH3ACACBCHRM2
SCHEMBL24639834 0.79 CHRM2 (0.34) NR1H2NR1H3HRH3ACACBCHRM2
SCHEMBL24640762 0.77 HRH3 (0.36) NR1H2NR1H3HRH3ACACBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed