SCHEMBL24639864

SCHEMBL24639864

CC(C)N1CCN2c3ncc(C(F)(F)F)cc3N(C3CC(F)(F)C3)C2C1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.33
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 2/20 0.33
ACACB O00763 2/20 0.33
TIPARP Q7Z3E1 4/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32
DRD3 P35462 1/20 0.32
HTR2B P41595 1/20 0.32
GAA P10253 1/20 0.31
ATM Q13315 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HCRTR1 O43613 1/20 0.31
SCN10A Q9Y5Y9 2/20 0.31
POLB P06746 1/20 0.31
CXCR3 P49682 1/20 0.30
OGA O60502 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24639836 0.88 HRH3 (0.35) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL24639834 0.88 CHRM2 (0.34) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL24639861 0.82 HRH3 (0.36) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL24639851 0.82 HRH3 (0.36) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL24639871 0.80 HRH3 (0.37) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL24639833 0.79 NR1H2 (0.37) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL31245432 0.79 HTR2C (0.36) HTR2BSCN10APOLB
SCHEMBL24639855 0.78 ACACB (0.40) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL24640155 0.77 CHRM2 (0.37) HRH3NR1H2NR1H3ACACBTIPARP
SCHEMBL26958078 0.77 CHRM2 (0.37) HRH3NR1H2NR1H3ACACBTIPARP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed