SCHEMBL24640233

SCHEMBL24640233

CC(C)N1CCN2c3ncc(C(F)(F)F)cc3NCC[C@H]2C1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TIPARP Q7Z3E1 6/20 0.49
HRH3 Q9Y5N1 4/20 0.35
ACACB O00763 2/20 0.35
PARP2 Q9UGN5 2/20 0.34
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
OGA O60502 3/20 0.33
CBLB Q13191 1/20 0.33
CHRM2 P08172 1/20 0.33
HTR1A P08908 1/20 0.33
DRD3 P35462 1/20 0.33
HTR2B P41595 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24640231 1.00 TIPARP (0.49) TIPARPHRH3ACACBPARP2NR1H2
SCHEMBL24640192 1.00 TIPARP (0.49) TIPARPHRH3ACACBPARP2NR1H2
SCHEMBL24640945 0.89 TIPARP (0.40) TIPARPHRH3ACACBNR1H2NR1H3
SCHEMBL26958125 0.86 TIPARP (0.47) TIPARPHRH3PARP2NR1H2NR1H3
SCHEMBL24640800 0.81 TIPARP (0.38) TIPARPHRH3ACACBNR1H2NR1H3
SCHEMBL24640054 0.81 TIPARP (0.38) TIPARPHRH3ACACBNR1H2NR1H3
SCHEMBL24640017 0.81 TIPARP (0.38) TIPARPHRH3ACACBNR1H2NR1H3
SCHEMBL24640184 0.80 POLB (0.38) TIPARPHRH3ACACBPARP2NR1H2
SCHEMBL24640243 0.80 POLB (0.38) TIPARPHRH3ACACBPARP2NR1H2
SCHEMBL24640193 0.80 POLB (0.38) TIPARPHRH3ACACBPARP2NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed