SCHEMBL24640938

SCHEMBL24640938

Cc1cnc2c(c1)OCC[C@@H]1CN(C)CCN21

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
SOS1 Q07889 1/20 0.37
TIPARP Q7Z3E1 11/20 0.35
PARP2 Q9UGN5 3/20 0.35
GRM5 P41594 4/20 0.35
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33
OPRK1 P41145 1/20 0.32
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24640360 1.00 HTR2A (0.38) HTR2AHTR2CHTR2BSOS1TIPARP
SCHEMBL24675032 0.87 HTR2A (0.34) HTR2AHTR2CHTR2BSOS1TIPARP
SCHEMBL24675019 0.87 HTR2A (0.34) HTR2AHTR2CHTR2BSOS1TIPARP
SCHEMBL24675018 0.87 HTR2A (0.34) HTR2AHTR2CHTR2BSOS1TIPARP
SCHEMBL24675045 0.86 HTR2A (0.37) HTR2AHTR2CHTR2BSOS1TIPARP
SCHEMBL24675043 0.86 HTR2A (0.37) HTR2AHTR2CHTR2BSOS1TIPARP
SCHEMBL24640827 0.84 NLRP3 (0.42) SOS1TIPARPPARP2GRM5CYP3A4
SCHEMBL24640620 0.84 TIPARP (0.47) HTR2AHTR2CHTR2BTIPARPPARP2
SCHEMBL24639353 0.84 SOS1 (0.41) SOS1TIPARPPARP2OPRK1
SCHEMBL24639358 0.84 SOS1 (0.41) SOS1TIPARPPARP2OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed