SCHEMBL2465035

SCHEMBL2465035

COc1ccnc(-c2cc(C3(c4cncnc4)N=C(N)c4ccccc43)ccc2F)c1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.47
KCNH2 Q12809 14/20 0.47
BACE2 Q9Y5Z0 5/20 0.41
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
REN P00797 1/20 0.37
CTSD P07339 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2465679 0.89 BACE1 (0.61) BACE1KCNH2BACE2
SCHEMBL2463159 0.80 BACE1 (0.63) BACE1KCNH2BACE2RENCTSD
SCHEMBL2086695 0.76 BACE1 (0.64) BACE1KCNH2BACE2RENCTSD
SCHEMBL2084717 0.75 BACE1 (0.71) BACE1KCNH2BACE2RENCTSD
SCHEMBL2461170 0.73 BACE1 (0.58) BACE1KCNH2BACE2RENCTSD
SCHEMBL2087395 0.72 BACE1 (0.60) BACE1KCNH2BACE2CTSD
SCHEMBL2086155 0.72 BACE1 (0.46) BACE1KCNH2BACE2CTSD
SCHEMBL3552580 0.72 BACE1 (0.55) BACE1KCNH2BACE2CTSD
SCHEMBL2086072 0.72 BACE1 (0.49) BACE1KCNH2BACE2CTSD
SCHEMBL3549935 0.71 BACE1 (0.74) BACE1KCNH2BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367814-A1 NEW COMPOUNDS 578 AstraZeneca AB (SE) 2011-09-28 EP disclosed
WO-2010056196-A1 NEW COMPOUNDS 578 ASTRAZENECA AB (SE) 2010-05-20 WO disclosed