SCHEMBL2463159

SCHEMBL2463159

COc1cc(C2(c3ccc(F)c(-c4cncnc4)c3)N=C(N)c3ccccc32)ccn1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.63
KCNH2 Q12809 14/20 0.63
BACE2 Q9Y5Z0 7/20 0.45
CTSD P07339 4/20 0.45
REN P00797 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2467948 0.89 BACE1 (0.80) BACE1KCNH2BACE2
SCHEMBL2084717 0.86 BACE1 (0.71) BACE1KCNH2BACE2CTSDREN
SCHEMBL2461925 0.85 BACE1 (0.75) BACE1KCNH2BACE2
SCHEMBL2086695 0.84 BACE1 (0.64) BACE1KCNH2BACE2CTSDREN
SCHEMBL2465035 0.80 BACE1 (0.47) BACE1KCNH2BACE2CTSDREN
SCHEMBL2086218 0.80 BACE1 (0.56) BACE1KCNH2BACE2CTSDREN
SCHEMBL8225712 0.79 BACE1 (0.58) BACE1KCNH2BACE2CTSDREN
SCHEMBL2462010 0.77 BACE1 (1.00) BACE1KCNH2BACE2
SCHEMBL2087779 0.77 BACE1 (0.58) BACE1KCNH2BACE2CTSD
SCHEMBL3356875 0.77 BACE1 (0.52) BACE1KCNH2BACE2CTSDREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367814-A1 NEW COMPOUNDS 578 AstraZeneca AB (SE) 2011-09-28 EP claimed
WO-2010056196-A1 NEW COMPOUNDS 578 ASTRAZENECA AB (SE) 2010-05-20 WO claimed