SCHEMBL24669355

SCHEMBL24669355

Cc1cc(C2=CCN(NC(=O)OC(C)(C)C)CC2)ccc1NC(=O)c1ccc(C2=CCNCC2)c(C)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.37
HTR1D P28221 2/20 0.34
HTR1B P28222 2/20 0.34
BTK Q06187 1/20 0.34
BRPF1 P55201 1/20 0.34
WDR5 P61964 1/20 0.33
MMP2 P08253 3/20 0.33
MMP3 P08254 3/20 0.33
NAMPT P43490 2/20 0.33
CCNT1 O60563 2/20 0.33
CDK9 P50750 2/20 0.33
SUCNR1 Q9BXA5 1/20 0.32
BRAF P15056 2/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671471 0.84 CSF1R (0.40) CSF1RBRPF1MMP2MMP3NAMPT
SCHEMBL29803364 0.83 QDPR (0.42) CSF1RBTKBRPF1NAMPTCCNT1
SCHEMBL29802842 0.80 NAMPT (0.52) WDR5NAMPTCCNT1CDK9
SCHEMBL24669309 0.80 NAMPT (0.52) WDR5NAMPTCCNT1CDK9
Trifluoroacetic Acid SCHEMBL29803809 0.80 P2RY14 (0.40) CSF1RBTKBRPF1NAMPTCCNT1
SCHEMBL29803575 0.76 NAMPT (0.40) MMP2MMP3NAMPTSUCNR1
SCHEMBL24669304 0.76 CCNT1 (0.47) CSF1RBTKBRPF1WDR5NAMPT
SCHEMBL29803667 0.76 CCNT1 (0.47) CSF1RBTKBRPF1WDR5NAMPT
SCHEMBL24670760 0.74 NAMPT (0.45) HTR1DNAMPT
SCHEMBL29803714 0.73 NAMPT (0.51) NAMPTCCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed