SCHEMBL24669403

SCHEMBL24669403

N=C(N)N1CC=C(c2ccc(C(=O)Nc3ccc4c(c3)CN(C(=N)N)CC4)cc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 8/20 0.69
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
PLAU P00749 3/20 0.47
NAMPT P43490 5/20 0.46
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803335 1.00 TMPRSS2 (0.69) TMPRSS2ITGB3ITGA2BPLAUNAMPT
SCHEMBL24671256 0.95 TMPRSS2 (0.67) TMPRSS2ITGB3ITGA2BNAMPT
SCHEMBL29802896 0.95 TMPRSS2 (0.67) TMPRSS2ITGB3ITGA2BNAMPT
SCHEMBL30180859 0.94 TMPRSS2 (0.66) TMPRSS2ITGB3ITGA2BNAMPT
SCHEMBL24891902 0.94 TMPRSS2 (0.66) TMPRSS2ITGB3ITGA2BNAMPT
SCHEMBL24891975 0.89 TMPRSS2 (0.80) TMPRSS2ITGB3ITGA2BPLAUNPC1
SCHEMBL29802903 0.89 TMPRSS2 (0.60) TMPRSS2PLAUNAMPTNPC1RAB9A
SCHEMBL24670202 0.89 TMPRSS2 (0.60) TMPRSS2PLAUNAMPTNPC1RAB9A
SCHEMBL24669348 0.88 TMPRSS2 (0.61) TMPRSS2ITGB3ITGA2BPLAUNAMPT
SCHEMBL29803057 0.88 TMPRSS2 (0.61) TMPRSS2ITGB3ITGA2BPLAUNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed