SCHEMBL24669348

SCHEMBL24669348

N=C(N)N1CC=C(c2ccc(C(=O)Nc3ccc4c(c3)CN(C(=N)N)CC4)cc2F)CC1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 8/20 0.61
NPC1 O15118 2/20 0.44
PLAU P00749 3/20 0.43
ITGB3 P05106 3/20 0.43
ITGA2B P08514 3/20 0.43
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NAMPT P43490 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803057 1.00 TMPRSS2 (0.61) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL24670135 0.95 TMPRSS2 (0.59) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL29802975 0.95 TMPRSS2 (0.59) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL29803214 0.91 TMPRSS2 (0.52) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL29803335 0.88 TMPRSS2 (0.69) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL24669403 0.88 TMPRSS2 (0.69) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL24669447 0.88 TMPRSS2 (0.48) TMPRSS2NPC1RAB9ASMN1; SMN2NAMPT
SCHEMBL29802849 0.87 TMPRSS2 (0.63) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL24671270 0.87 TMPRSS2 (0.52) TMPRSS2NPC1PLAUITGB3ITGA2B
SCHEMBL24670643 0.87 TMPRSS2 (0.52) TMPRSS2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed