SCHEMBL24669484

SCHEMBL24669484

O=C(Nc1cc(F)c(Br)c(F)c1)c1ccc(Br)c(F)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.59
MAPT P10636 2/20 0.47
KCNQ3 O43525 6/20 0.46
KCNQ2 O43526 6/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
KCNQ5 Q9NR82 3/20 0.46
KCNE1 P15382 3/20 0.44
KCNQ1 P51787 3/20 0.44
XBP1 P17861 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
RARA P10276 1/20 0.43
RARB P10826 1/20 0.43
RARG P13631 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24669338 0.90 MAOB (0.70) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL29803408 0.90 MAOB (0.70) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL24670951 0.90 MAOB (0.53) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL24671323 0.86 MAOB (0.65) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL24670922 0.84 TP53 (0.63) MAOBMAPTNPC1RAB9AMEN1
SCHEMBL24670735 0.80 MAOB (0.62) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL24670043 0.80 MAPT (0.77) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL29803768 0.80 MAPT (0.77) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL24670851 0.80 MAOB (0.59) MAOBMAPTKCNQ3KCNQ2NPC1
SCHEMBL29803287 0.80 MAOB (0.59) MAOBMAPTKCNQ3KCNQ2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed