SCHEMBL24669727

SCHEMBL24669727

NS(=O)(=O)c1cc(CCCn2cnc3c(NCc4ccccc4)nc(F)nc32)on1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.47
PDE5A O76074 2/20 0.47
CDK2 P24941 2/20 0.46
CTSL P07711 7/20 0.45
TMIGD3 P0DMS9 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
CCNA2 P20248 1/20 0.43
CCNA1 P78396 1/20 0.43
CACNA1B Q00975 1/20 0.43
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
CTSB P07858 1/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24669726 0.85 CDK2 (0.67) CDK1CDK2CCNA2CCNA1CACNA1B
SCHEMBL24669716 0.84 CDK1 (0.48) CDK1PDE5ACDK2CTSLTMIGD3
SCHEMBL24668665 0.82 CTSL (0.46) CDK1PDE5ACDK2CTSLTMIGD3
SCHEMBL24668664 0.82 PDE5A (0.47) CDK1PDE5ACDK2CTSLTMIGD3
SCHEMBL24670389 0.81 CTSL (0.47) CDK1PDE5ACDK2CTSLTMIGD3
SCHEMBL24668634 0.80 PDE5A (0.47) CDK1PDE5ACDK2CTSLTMIGD3
SCHEMBL24669107 0.78 CTSL (0.47) CDK1PDE5ACDK2CTSLTMIGD3
SCHEMBL24670403 0.77 PDE5A (0.51) CDK1PDE5ACDK2CTSLTMIGD3
SCHEMBL17450142 0.76 CTSL (0.67) CDK1CDK2CTSLTMIGD3ADORA2A
SCHEMBL17450124 0.74 CDK1 (0.72) CDK1CDK2CTSLTMIGD3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187693-A1 COVALENT CDK2-BINDING COMPOUNDS FOR THERAPEUTIC PURPOSES UMBRA THERAPEUTICS INC. (US) 2022-09-09 WO disclosed