SCHEMBL24670077

SCHEMBL24670077

CSc1ncc(CO)c(NCc2ccc(-c3ncc(Br)o3)cc2)n1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.53
AGTR1 P30556 5/20 0.41
AGTR2 P50052 5/20 0.41
PPARG P37231 2/20 0.36
RXFP1 Q9HBX9 3/20 0.35
THRB P10828 2/20 0.35
USP1 O94782 1/20 0.34
WDR48 Q8TAF3 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK5 Q00535 1/20 0.34
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670411 0.86 HTT (0.53) HTTAGTR1AGTR2PPARGRXFP1
SCHEMBL24670075 0.83 CA1 (0.39) HTTPPARGRXFP1THRBUSP1
SCHEMBL4712339 0.77 HTT (0.76) HTTCCNE1CDK2POLBLMNA
SCHEMBL24669161 0.74 HTT (0.52) HTTAGTR1AGTR2PPARGRXFP1
SCHEMBL14914628 0.72 HTT (0.65) HTTPPARGPOLBLMNA
SCHEMBL24669149 0.71 HTT (0.56) HTTAGTR1AGTR2RXFP1THRB
SCHEMBL24669124 0.71 HTT (0.50) HTTAGTR1AGTR2CCNE1CDK2
SCHEMBL24668698 0.71 HTT (0.50) HTTAGTR1AGTR2RXFP1THRB
SCHEMBL1521623 0.70 HTT (0.55) HTTAGTR1AGTR2THRBPOLB
SCHEMBL24670415 0.69 CA1 (0.42) HTTPPARGRXFP1THRBUSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187693-A1 COVALENT CDK2-BINDING COMPOUNDS FOR THERAPEUTIC PURPOSES UMBRA THERAPEUTICS INC. (US) 2022-09-09 WO disclosed