SCHEMBL24670075

SCHEMBL24670075

CSc1ncc(C=O)c(NCc2ccc(-c3ncc(Br)o3)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA13 Q8N1Q1 2/20 0.39
PPARG P37231 3/20 0.36
HTT P42858 1/20 0.35
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK5 Q00535 1/20 0.34
RXFP1 Q9HBX9 3/20 0.33
THRB P10828 2/20 0.33
AKT1 P31749 2/20 0.33
AKT2 P31751 2/20 0.33
USP1 O94782 1/20 0.32
WDR48 Q8TAF3 1/20 0.32
POLB P06746 1/20 0.31
TP53 P04637 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ABL1 P00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670415 0.86 CA1 (0.42) CA1CA2CA7CA13PPARG
SCHEMBL24670077 0.83 HTT (0.53) PPARGHTTCCNE1CDK2CDK5
SCHEMBL2554057 0.78 PPARG (0.51) CA1CA2CA7CA13PPARG
SCHEMBL4712462 0.77 HTT (0.51) CA1CA2CA7CA13HTT
SCHEMBL24669163 0.74 CA1 (0.39) CA1CA2CA7CA13PPARG
SCHEMBL14914225 0.72 PPARG (0.53) CA1CA2CA7CA13PPARG
SCHEMBL24669160 0.72 CA1 (0.52) CA1CA2CA7CA13HTT
SCHEMBL24670094 0.72 CA1 (0.49) CA1CA2CA7CA13PPARG
SCHEMBL24668699 0.71 CA2 (0.47) CA1CA2CA7CA13HTT
SCHEMBL24669128 0.71 CA1 (0.52) CA1CA2CA7CA13HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187693-A1 COVALENT CDK2-BINDING COMPOUNDS FOR THERAPEUTIC PURPOSES UMBRA THERAPEUTICS INC. (US) 2022-09-09 WO disclosed