SCHEMBL24670094

SCHEMBL24670094

CSc1ncc(C=O)c(NCc2ccc(CCCS(N)(=O)=O)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 11/20 0.49
CA2 P00918 11/20 0.49
CA13 Q8N1Q1 5/20 0.49
CA7 P43166 5/20 0.49
HTT P42858 1/20 0.35
CA9 Q16790 5/20 0.34
CA12 O43570 1/20 0.34
CA4 P22748 1/20 0.34
PPARG P37231 3/20 0.34
STAT6 P42226 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670432 0.90 CA1 (0.44) CA1CA2CA13CA7HTT
SCHEMBL16415327 0.83 CA1 (0.41) CA1CA2CA13CA7HTT
SCHEMBL2554057 0.79 PPARG (0.51) CA1CA2CA13CA7HTT
SCHEMBL4712462 0.78 HTT (0.51) CA1CA2CA13CA7HTT
SCHEMBL24669160 0.77 CA1 (0.52) CA1CA2CA13CA7HTT
SCHEMBL24669128 0.76 CA1 (0.52) CA1CA2CA13CA7HTT
SCHEMBL24668699 0.76 CA2 (0.47) CA1CA2CA13CA7HTT
SCHEMBL24669602 0.75 CA1 (0.51) CA1CA2CA13CA7HTT
SCHEMBL24670428 0.75 HTT (0.49) CA1CA2CA13CA7HTT
SCHEMBL24669065 0.74 CA1 (0.43) CA1CA2CA13CA7HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187693-A1 COVALENT CDK2-BINDING COMPOUNDS FOR THERAPEUTIC PURPOSES UMBRA THERAPEUTICS INC. (US) 2022-09-09 WO disclosed