SCHEMBL24670296

SCHEMBL24670296

CC(C)(C)OC(=O)NCCc1ccc(NC(=O)c2ccc(C3=CCN(C(=O)OC(C)(C)C)CC3)cc2F)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.50
WNT3A P56704 1/20 0.44
LIPC P11150 1/20 0.40
LIPG Q9Y5X9 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
KIT P10721 2/20 0.39
CDK7 P50613 1/20 0.39
CDK13 Q14004 1/20 0.39
CDK12 Q9NYV4 1/20 0.39
MCHR1 Q99705 1/20 0.39
GRM5 P41594 5/20 0.39
GRM1 Q13255 5/20 0.39
WDR5 P61964 1/20 0.38
SOS1 Q07889 1/20 0.38
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
ESRRG P62508 1/20 0.37
PTGER4 P35408 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803379 0.88 NAMPT (0.55) NAMPTWNT3ALIPCLIPGKIT
SCHEMBL24671383 0.85 NAMPT (0.40) NAMPTWNT3AMCHR1CCNT1CDK9
SCHEMBL24671384 0.85 NAMPT (0.40) NAMPTWNT3AMCHR1CCNT1CDK9
SCHEMBL24891933 0.84 NAMPT (0.55) NAMPTWNT3ALIPCLIPGKIT
SCHEMBL24892373 0.84 NAMPT (0.55) NAMPTWNT3ALIPCLIPGKIT
SCHEMBL29803362 0.84 NAMPT (0.48) NAMPTWNT3AKITMCHR1GRM5
SCHEMBL24671267 0.83 NAMPT (0.49) NAMPTWNT3ALIPCLIPGKIT
SCHEMBL24669471 0.82 NAMPT (0.53) NAMPTWNT3ATLR7CDK7CDK13
SCHEMBL24670609 0.81 NAMPT (0.52) NAMPTWNT3ATLR7CDK7CDK13
SCHEMBL29803508 0.81 NAMPT (0.52) NAMPTWNT3ATLR7CDK7CDK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed