SCHEMBL24670487

SCHEMBL24670487

CC(C)(C)OC(=O)N1CC=C(c2ccc(NC(=O)c3cc(C4=CCN(C(=O)OC(C)(C)C)CC4)co3)cc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 6/20 0.61
WNT3A P56704 1/20 0.47
CDK7 P50613 1/20 0.46
CDK13 Q14004 1/20 0.46
CDK12 Q9NYV4 1/20 0.46
PTPN2 P17706 1/20 0.45
PTPN1 P18031 1/20 0.45
PTPN6 P29350 1/20 0.45
PDK4 Q16654 1/20 0.45
JAK1 P23458 1/20 0.43
KIT P10721 1/20 0.43
GRM1 Q13255 7/20 0.43
GRM5 P41594 6/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24669214 0.92 NAMPT (0.52) NAMPTWNT3AGRM1GRM5
SCHEMBL24669868 0.89 NAMPT (0.49) NAMPTWNT3ACDK7CDK13CDK12
SCHEMBL29803286 0.89 NAMPT (0.49) NAMPTWNT3ACDK7CDK13CDK12
SCHEMBL24670536 0.88 NAMPT (0.47) NAMPTWNT3ACDK7CDK13CDK12
SCHEMBL24671065 0.87 NAMPT (0.49) NAMPTWNT3ACDK7CDK13CDK12
SCHEMBL24669237 0.84 NAMPT (0.50) NAMPTWNT3ACDK7CDK13CDK12
SCHEMBL24670493 0.84 NAMPT (0.46) NAMPTWNT3A
SCHEMBL24670496 0.84 NAMPT (0.46) NAMPTWNT3A
SCHEMBL29803394 0.82 NAMPT (0.48) NAMPTWNT3ACDK7CDK13CDK12
Lithium Ion SCHEMBL29803642 0.82 NAMPT (0.48) NAMPTCDK7CDK13CDK12PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed