SCHEMBL24671065

SCHEMBL24671065

CC(C)(C)OC(=O)N1CC=C(c2ccc(NC(=O)c3cc(C4=CCN(C(=O)OC(C)(C)C)CC4)co3)nc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.49
CDK7 P50613 1/20 0.46
CDK13 Q14004 1/20 0.46
CDK12 Q9NYV4 1/20 0.46
WNT3A P56704 1/20 0.46
CYP11B2 P19099 1/20 0.45
JAK1 P23458 1/20 0.44
GRM5 P41594 2/20 0.43
GRM1 Q13255 2/20 0.43
EED O75530 1/20 0.42
RBBP4 Q09028 1/20 0.42
SUZ12 Q15022 1/20 0.42
EZH2 Q15910 1/20 0.42
ATR Q13535 1/20 0.42
KIT P10721 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670487 0.87 NAMPT (0.61) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL29803615 0.85 NAMPT (0.44) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24670527 0.85 NAMPT (0.44) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24669270 0.85 NAMPT (0.44) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL22165464 0.84 NAMPT (0.56) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24670528 0.83 NAMPT (0.46) NAMPT
SCHEMBL24669665 0.81 NAMPT (0.48) NAMPTCDK7CDK13CDK12WNT3A
Trifluoroacetic Acid SCHEMBL29803709 0.80 NAMPT (0.43) NAMPT
SCHEMBL29803476 0.80 NAMPT (0.49) NAMPTCDK7CDK13CDK12WNT3A
SCHEMBL24669237 0.80 NAMPT (0.50) NAMPTCDK7CDK13CDK12WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed