SCHEMBL24670530

SCHEMBL24670530

O=C(Nc1ccc(Br)s1)c1ccc(I)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
TP53 P04637 2/20 0.45
NFKB1 P19838 2/20 0.45
NFKB2 Q00653 2/20 0.45
RELA Q04206 2/20 0.45
TRPV1 Q8NER1 3/20 0.44
ADORA3 P0DMS8 2/20 0.40
ABL1 P00519 1/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
LMNA P02545 2/20 0.40
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 1/20 0.39
RNASEH1 O60930 1/20 0.39
TPMT P51580 1/20 0.38
GSK3B P49841 1/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670532 0.83 NPC1 (0.53) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL26983703 0.72 DAO (0.48) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL7057048 0.71 GAA (0.43) MAPTSMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL11191679 0.71 HSD17B10 (0.72) MAPTSMN1; SMN2NPC1RAB9AABL1
SCHEMBL21653125 0.70 BRD4 (0.40) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL3674376 0.70 TRPV1 (0.76) SMN1; SMN2NPC1RAB9ATP53TRPV1
SCHEMBL21694316 0.69 HDAC6 (0.60) TPMTCA1CA2ALOX15HSD17B10
SCHEMBL16482164 0.69 IL2 (0.54) SMN1; SMN2RAB9ATP53KMT2AMEN1
SCHEMBL7103601 0.69 MEN1 (0.68) NPC1RAB9ATP53TRPV1KMT2A
SCHEMBL27989047 0.68 GAA (0.45) MAPTSMN1; SMN2NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed