SCHEMBL24670587

SCHEMBL24670587

COc1cc(NC(=O)c2ccc(C3=CCN(C(=O)OC(C)(C)C)CC3)s2)ccc1C1=CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.46
PDK4 Q16654 1/20 0.44
GRM5 P41594 2/20 0.43
GRM1 Q13255 2/20 0.43
JAK1 P23458 1/20 0.43
IMPDH2 P12268 2/20 0.41
KIT P10721 1/20 0.41
SCN9A Q15858 2/20 0.41
F13A1 P00488 1/20 0.40
TGM2 P21980 1/20 0.40
TGM1 P22735 1/20 0.40
TRPV1 Q8NER1 2/20 0.40
PDE10A Q9Y233 1/20 0.40
HTR6 P50406 1/20 0.40
WNT3A P56704 2/20 0.39
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803262 1.00 NAMPT (0.46) NAMPTPDK4GRM5GRM1JAK1
SCHEMBL29803799 0.89 NAMPT (0.47) NAMPTPDK4GRM5GRM1JAK1
SCHEMBL29803594 0.89 NAMPT (0.47) NAMPTPDK4GRM5GRM1JAK1
SCHEMBL24669259 0.89 NAMPT (0.47) NAMPTPDK4GRM5GRM1JAK1
SCHEMBL24671091 0.89 NAMPT (0.47) NAMPTPDK4GRM5GRM1JAK1
SCHEMBL24670551 0.86 TMPRSS2 (0.44) IMPDH2TRPV1WNT3A
SCHEMBL29803002 0.86 TMPRSS2 (0.44) IMPDH2TRPV1WNT3A
SCHEMBL24670469 0.86 NAMPT (0.49) NAMPTPDK4GRM5GRM1JAK1
SCHEMBL29803715 0.86 NAMPT (0.49) NAMPTPDK4GRM5GRM1JAK1
SCHEMBL29803749 0.86 IMPDH2 (0.37) NAMPTPDK4GRM5GRM1JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed