SCHEMBL24670973

SCHEMBL24670973

CC(C)(C)OC(=O)N1CC=C(c2ccc(NC(=O)c3ccc(C4=CCB(C#N)CC4)cc3F)cc2Cl)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.43
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
MAPT P10636 5/20 0.39
HTT P42858 3/20 0.39
KMT2A Q03164 2/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PDK4 Q16654 1/20 0.38
WDR5 P61964 2/20 0.37
CDK7 P50613 1/20 0.37
CDK13 Q14004 1/20 0.37
CDK12 Q9NYV4 1/20 0.37
NPSR1 Q6W5P4 2/20 0.37
CNR1 P21554 1/20 0.37
GPR35 Q9HC97 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803557 0.91 NAMPT (0.51) NAMPTALDH1A1TRPV1MAPTHTT
SCHEMBL24669521 0.91 NAMPT (0.51) NAMPTALDH1A1TRPV1MAPTHTT
SCHEMBL24671313 0.85 WDR5 (0.43) NAMPTPDK4WDR5CDK7CDK13
SCHEMBL24669471 0.83 NAMPT (0.53) NAMPTPDK4WDR5CDK7CDK13
SCHEMBL24669429 0.82 PDK4 (0.39) NAMPTMAPTPDK4WDR5JAK1
SCHEMBL24669408 0.81 NAMPT (0.50) NAMPTMAPTPDK4WDR5CDK7
SCHEMBL24670598 0.79 PDK4 (0.39) NAMPTPDK4WDR5JAK1GRM5
SCHEMBL24670300 0.78 NAMPT (0.39) NAMPTALDH1A1L3MBTL1TRPV1MAPT
SCHEMBL24669509 0.78 NAMPT (0.39) NAMPTALDH1A1L3MBTL1TRPV1MAPT
SCHEMBL29803520 0.78 NAMPT (0.39) NAMPTALDH1A1L3MBTL1TRPV1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed