SCHEMBL24671224

SCHEMBL24671224

CC(C)(C)OC(=O)/N=C(\NC(=O)OC(C)(C)C)N1CC=C(c2ccc(N)cc2F)CC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.39
PDK4 Q16654 1/20 0.38
CDK9 P50750 3/20 0.36
GRM5 P41594 5/20 0.36
GRM1 Q13255 5/20 0.36
NAMPT P43490 1/20 0.35
JAK1 P23458 1/20 0.35
CCNT1 O60563 1/20 0.34
HTR6 P50406 1/20 0.34
WDR5 P61964 2/20 0.34
SCN9A Q15858 2/20 0.33
TNF P01375 1/20 0.33
EED O75530 1/20 0.33
RBBP4 Q09028 1/20 0.33
SUZ12 Q15022 1/20 0.33
EZH2 Q15910 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670577 0.91 PDK4 (0.39) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24671139 0.90 NR1H2 (0.40) NR1H2PDK4CDK9GRM5GRM1
SCHEMBL24670136 0.90 NR1H2 (0.40) NR1H2PDK4CDK9GRM5GRM1
SCHEMBL24670675 0.89 NR1H2 (0.38) NR1H2PDK4CDK9GRM5GRM1
SCHEMBL24670618 0.89 NR1H2 (0.39) NR1H2PDK4CDK9GRM5GRM1
SCHEMBL24669395 0.88 NR1H2 (0.39) NR1H2PDK4CDK9GRM5GRM1
SCHEMBL24670250 0.88 GRM1 (0.36) NR1H2PDK4CDK9GRM5GRM1
SCHEMBL24671099 0.88 PDK4 (0.38) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24669650 0.86 PDK4 (0.35) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24670260 0.86 NR1H2 (0.37) NR1H2PDK4CDK9GRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed