SCHEMBL24670577

SCHEMBL24670577

Cc1ccc(C2=CCN(C(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)CC2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.39
CDK9 P50750 3/20 0.37
GRM5 P41594 5/20 0.37
GRM1 Q13255 5/20 0.37
NAMPT P43490 1/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
GABRE P78334 1/20 0.36
GABRA6 Q16445 1/20 0.36
GABRG1 Q8N1C3 1/20 0.36
GABRG3 Q99928 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671224 0.91 NR1H2 (0.39) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24669345 0.90 PDK4 (0.40) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24671099 0.89 PDK4 (0.38) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24670620 0.89 PDK4 (0.39) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL27025875 0.88 CDK9 (0.37) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24670284 0.87 SCN9A (0.38) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24669650 0.86 PDK4 (0.35) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL29803193 0.86 NAMPT (0.40) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL27025948 0.86 TRPV1 (0.39) PDK4CDK9GRM5GRM1NAMPT
SCHEMBL24670250 0.86 GRM1 (0.36) PDK4CDK9GRM5GRM1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed