SCHEMBL24671346

SCHEMBL24671346

CC(C)NC(=O)c1ccc(C2=CCNCC2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
NPSR1 Q6W5P4 1/20 0.43
CCNT1 O60563 3/20 0.41
CDK9 P50750 3/20 0.41
MLYCD O95822 1/20 0.41
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41
PDK2 Q15119 1/20 0.40
HTR2C P28335 2/20 0.39
P2RY14 Q15391 1/20 0.39
WDR5 P61964 2/20 0.39
BRPF1 P55201 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670266 0.85 CCNT1 (0.52) NPSR1CCNT1CDK9MLYCDROCK1
SCHEMBL31702208 0.81 PDE3B (0.47) PDE3BPDE3ACCNT1CDK9PDK2
SCHEMBL29803919 0.80 CCNT1 (0.44) PDE3BPDE3ANPSR1CCNT1CDK9
SCHEMBL29803888 0.78 CCNT1 (0.46) PDE3BPDE3ANPSR1CCNT1CDK9
Trifluoroacetic Acid SCHEMBL29803720 0.77 CCNT1 (0.41) PDE3BPDE3ANPSR1CCNT1CDK9
SCHEMBL24670780 0.74 CCNT1 (0.39) CCNT1CDK9ROCK2ROCK1
SCHEMBL24670935 0.74 CCNT1 (0.39) CCNT1CDK9HTR2CBRPF1
SCHEMBL5536591 0.74 PDE3B (0.52) PDE3BPDE3AHTR2C
SCHEMBL24671030 0.72 CCNT1 (0.47) CCNT1CDK9WDR5BRPF1
SCHEMBL24670925 0.72 CCNT1 (0.41) CCNT1CDK9ROCK2ROCK1WDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed