SCHEMBL24671439

SCHEMBL24671439

Cc1c(NC(=O)c2ccc(C3=CCN(C(=O)OC(C)(C)C)CC3)c(F)c2)ccc(C2=CCN(C(=O)OC(C)(C)C)CC2)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.46
WDR5 P61964 2/20 0.45
PDK4 Q16654 1/20 0.44
NAMPT P43490 1/20 0.44
DGAT2 Q96PD7 1/20 0.44
CDK9 P50750 3/20 0.43
CCNT1 O60563 1/20 0.43
JAK1 P23458 1/20 0.43
GRM5 P41594 7/20 0.42
GRM1 Q13255 7/20 0.42
CNR1 P21554 1/20 0.42
HTR6 P50406 1/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803533 0.93 WDR5 (0.47) SCN9AWDR5PDK4NAMPTDGAT2
SCHEMBL24669512 0.92 SCN9A (0.46) SCN9AWDR5PDK4NAMPTCDK9
SCHEMBL24669486 0.88 SCN9A (0.47) SCN9AWDR5PDK4NAMPTDGAT2
SCHEMBL29803593 0.88 NAMPT (0.49) SCN9AWDR5PDK4NAMPTDGAT2
SCHEMBL24669316 0.88 WDR5 (0.48) SCN9AWDR5PDK4NAMPTDGAT2
SCHEMBL29803452 0.88 WDR5 (0.48) SCN9AWDR5PDK4NAMPTDGAT2
SCHEMBL24670264 0.87 WDR5 (0.49) SCN9AWDR5PDK4NAMPTDGAT2
SCHEMBL24670616 0.87 NAMPT (0.49) SCN9AWDR5PDK4NAMPTCDK9
SCHEMBL24670846 0.86 WDR5 (0.35) SCN9AWDR5PDK4NAMPTDGAT2
SCHEMBL29803745 0.86 WDR5 (0.35) SCN9AWDR5PDK4NAMPTDGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed