SCHEMBL24671458

SCHEMBL24671458

COc1cc(NC(=O)c2ccc(Br)cc2)ccc1Br

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.63
RAB9A P51151 5/20 0.61
TP53 P04637 4/20 0.61
NPC1 O15118 4/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
ALDH1A1 P00352 1/20 0.61
GRM4 Q14833 1/20 0.60
MAPT P10636 5/20 0.55
POLB P06746 3/20 0.54
KDR P35968 1/20 0.54
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
STAT1 P42224 1/20 0.53
MAPK1 P28482 1/20 0.52
ALOX15 P16050 1/20 0.51
SAE1 Q9UBE0 1/20 0.51
UBA2 Q9UBT2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256379 0.90 NPC1 (0.76) ABCB1RAB9ATP53NPC1SMN1; SMN2
SCHEMBL24670914 0.86 HTR1D (0.65) ABCB1RAB9ATP53NPC1SMN1; SMN2
SCHEMBL29803730 0.85 GRM4 (0.56) RAB9ATP53NPC1SMN1; SMN2ALDH1A1
SCHEMBL24669380 0.85 GRM4 (0.56) RAB9ATP53NPC1SMN1; SMN2ALDH1A1
SCHEMBL24670802 0.85 MAPT (0.67) RAB9ATP53NPC1SMN1; SMN2ALDH1A1
SCHEMBL10035062 0.84 ABCB1 (0.55) ABCB1RAB9ATP53NPC1SMN1; SMN2
SCHEMBL24670251 0.83 POLB (0.56) ABCB1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL24670265 0.83 GRM4 (0.55) RAB9ATP53NPC1SMN1; SMN2ALDH1A1
SCHEMBL24670737 0.83 HTR1D (0.61) ABCB1RAB9ATP53NPC1SMN1; SMN2
SCHEMBL29803389 0.83 HTR1D (0.61) ABCB1RAB9ATP53NPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed