SCHEMBL24672390

SCHEMBL24672390

NC(=O)c1c[nH]c2nccc(Cl)c12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 3/20 0.62
LRRK2 Q5S007 2/20 0.62
CDK2 P24941 2/20 0.62
CDK9 P50750 2/20 0.62
CDK5 Q00535 2/20 0.62
AURKB Q96GD4 2/20 0.62
AXL P30530 2/20 0.62
PRKCI P41743 2/20 0.62
MAP2K1 Q02750 2/20 0.62
CDC7 O00311 1/20 0.62
PLK4 O00444 1/20 0.62
CHEK1 O14757 1/20 0.62
MAPK13 O15264 1/20 0.62
PDPK1 O15530 1/20 0.62
DAPK3 O43293 1/20 0.62
DYRK3 O43781 1/20 0.62
ROCK2 O75116 1/20 0.62
PRKD3 O94806 1/20 0.62
MAP4K4 O95819 1/20 0.62
ABL1 P00519 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30668776 1.00 CDK8 (0.62) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL30122008 0.85 CSNK2A1 (0.52) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL17818839 0.85 CSNK2A1 (0.52) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL2888458 0.84 CYP3A4 (0.60) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL1839435 0.84 LRRK2 (0.51) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL17818802 0.81 NR4A2 (0.58) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL20744099 0.81 LRRK2 (0.49) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL23610513 0.81 PRKCI (0.45) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL27019698 0.80 CDK2 (0.54) CDK8LRRK2CDK2CDK9CDK5
SCHEMBL21678754 0.79 LRRK2 (0.47) CDK8LRRK2CDK2CDK9CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111278840-B Pyrrolo [2,3-B ] pyridine compounds and their use for the treatment of cancer 癌症研究科技有限公司 2023-11-17 CN disclosed
US-11447505-B1 Pyrrolo[2,3-b]pyridine compounds and their use in the treatment of cancer CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2022-09-20 US disclosed
US-11447505-B1 Pyrrolo[2,3-b]pyridine compounds and their use in the treatment of cancer CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2022-09-20 US disclosed
CN-111278840-A Pyrrolo [2, 3-B ] pyridine compounds and their use for treating cancer 癌症研究科技有限公司 2020-06-12 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11447505-B1 Pyrrolo[2,3-b]pyridine compounds and their use in the treatment of cancer PDXK, CCNK, CDC42BPB CDK8 308/4885LRRK2 899/4885CDK2 71/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.