SCHEMBL24676593

SCHEMBL24676593

CN(C)Cc1nc(C(F)(F)F)c(-c2nc(NC3CCN(C(=O)OC(C)(C)C)CC3)ncc2F)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK2 Q92630 6/20 0.43
IDH1 O75874 1/20 0.41
IDH2 P48735 1/20 0.41
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
CCND3 P30281 1/20 0.41
CDK6 Q00534 1/20 0.41
CDK2 P24941 2/20 0.39
CDK1 P06493 1/20 0.39
GPR119 Q8TDV5 2/20 0.39
MAPK1 P28482 2/20 0.39
SYK P43405 1/20 0.39
CCNT1 O60563 1/20 0.39
ALDH1A1 P00352 2/20 0.38
CCNA2 P20248 1/20 0.38
KDM1A O60341 1/20 0.38
EHMT2 Q96KQ7 1/20 0.38
RCOR1 Q9UKL0 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676598 0.92 DYRK2 (0.44) DYRK2IDH1IDH2CDK4CCND1
SCHEMBL24676684 0.90 CDK2 (0.43) DYRK2IDH1CDK4CCND1CCND3
SCHEMBL24676928 0.89 CDK4 (0.36) DYRK2IDH1IDH2CDK4CCND1
SCHEMBL29754914 0.89 CDK4 (0.36) DYRK2IDH1IDH2CDK4CCND1
SCHEMBL24676591 0.88 DYRK2 (0.41) DYRK2IDH1IDH2CDK4CCND1
SCHEMBL24676105 0.84 CDK2 (0.36) CDK4CCND1CCND3CDK6CDK2
SCHEMBL24676566 0.84 CCNE1 (0.45) CDK4CCND1CCND3CDK6CDK2
SCHEMBL29754806 0.84 CDK2 (0.54) CDK4CCND1CCND3CDK6CDK2
SCHEMBL24676765 0.84 CDK2 (0.54) CDK4CCND1CCND3CDK6CDK2
SCHEMBL24676103 0.84 CCNE1 (0.47) CDK4CCND1CCND3CDK6CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed