SCHEMBL24676800

SCHEMBL24676800

CC(C)Nc1nc(C(F)(F)F)c(-c2ccnc(NC3CCN(S(C)(=O)=O)CC3)n2)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 4/20 0.53
CDK2 P24941 14/20 0.49
CCND1 P24385 9/20 0.49
CDK6 Q00534 9/20 0.49
CCNA2 P20248 8/20 0.49
CDK4 P11802 8/20 0.49
CDK1 P06493 8/20 0.49
CCNB1 P14635 8/20 0.49
CCND3 P30281 7/20 0.49
CDK7 P50613 7/20 0.49
CCNH P51946 7/20 0.49
CCNT1 O60563 6/20 0.49
CDK9 P50750 6/20 0.49
CCNE1 P24864 6/20 0.46
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46
MAPK10 P53779 1/20 0.46
CCNA1 P78396 2/20 0.45
IDH1 O75874 1/20 0.43
IDH2 P48735 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24676922 0.91 CDK2 (0.58) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL24676704 0.90 IKBKB (0.56) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL29755006 0.90 IKBKB (0.56) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL24675961 0.85 IKBKB (0.58) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL24676792 0.83 CDK2 (0.54) CDK2CCND1CDK6CCNA2CDK4
SCHEMBL29754874 0.83 IKBKB (0.54) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL24675988 0.83 IKBKB (0.54) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL24676930 0.82 IKBKB (0.52) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL29754851 0.82 IKBKB (0.52) IKBKBCDK2CCND1CDK6CCNA2
SCHEMBL24677023 0.81 IKBKB (0.52) IKBKBCDK2CCND1CDK6CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed