SCHEMBL24676855

SCHEMBL24676855

CSN1CCC(Nc2ncc(C#N)c(-c3sc(C4CC4)nc3C(F)(F)F)n2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 16/20 0.39
CCNE1 P24864 13/20 0.39
CCNT1 O60563 11/20 0.39
CDK9 P50750 11/20 0.39
CDK7 P50613 10/20 0.39
CCNH P51946 10/20 0.39
CDK1 P06493 9/20 0.39
CCNB1 P14635 9/20 0.39
MNAT1 P51948 8/20 0.39
CDK4 P11802 7/20 0.39
CCND1 P24385 7/20 0.39
CCND3 P30281 7/20 0.39
CDK6 Q00534 7/20 0.39
JUN P05412 1/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
CCNA2 P20248 2/20 0.34
CCNK O75909 4/20 0.32
CDK12 Q9NYV4 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24677062 0.87 CDK2 (0.38) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24676822 0.86 CDK2 (0.41) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL29754876 0.86 CCNE1 (0.49) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24676854 0.86 CCNE1 (0.49) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24676017 0.85 CCND1 (0.39) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24676938 0.84 CDK2 (0.39) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24677066 0.84 CDK4 (0.37) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24676853 0.84 CDK4 (0.36) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24677074 0.82 CDK2 (0.38) CDK2CCNE1CCNT1CDK9CDK7
SCHEMBL24676957 0.81 CDK4 (0.38) CDK2CCNE1CCNT1CDK9CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed