Trimecaine

Trimecaine

SCHEMBL24692

CCN(CC)CC(=O)Nc1c(C)cc(C)cc1C

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.97
TSHR P16473 2/20 0.72
RAB9A P51151 1/20 0.72
ALDH1A1 P00352 5/20 0.71
MAPT P10636 4/20 0.71
LMNA P02545 3/20 0.71
CYP3A4 P08684 1/20 0.71
MAPK1 P28482 1/20 0.71
MC4R P32245 1/20 0.71
SCN4A P35499 1/20 0.71
MC3R P41968 1/20 0.71
HTR3A P46098 1/20 0.71
SCN5A Q14524 1/20 0.71
SCN9A Q15858 1/20 0.71
SCN3A Q9NY46 1/20 0.71
GAA P10253 3/20 0.69
BLM P54132 1/20 0.69
NPSR1 Q6W5P4 1/20 0.56
POLB P06746 3/20 0.50
NR4A1 P22736 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trimecaine SCHEMBL1651359 0.98 HPGD (1.00) HPGDTSHRRAB9AALDH1A1MAPT
Trimecaine SCHEMBL28896832 0.98 HPGD (0.94) HPGDTSHRRAB9AALDH1A1MAPT
Trimecaine SCHEMBL28896992 0.97 HPGD (0.97) HPGDTSHRRAB9AALDH1A1MAPT
Trimecaine SCHEMBL28896917 0.97 HPGD (0.97) HPGDTSHRRAB9AALDH1A1MAPT
Trimecaine SCHEMBL28896834 0.97 HPGD (0.97) HPGDTSHRRAB9AALDH1A1MAPT
SCHEMBL21261833 0.88 HPGD (0.77) HPGDTSHRRAB9AALDH1A1MAPT
SCHEMBL2615417 0.87 HPGD (0.74) HPGDTSHRRAB9AALDH1A1MAPT
SCHEMBL2615419 0.87 HPGD (0.74) HPGDTSHRRAB9AALDH1A1MAPT
SCHEMBL11654851 0.87 HPGD (0.74) HPGDTSHRRAB9AALDH1A1MAPT
SCHEMBL10640761 0.85 HPGD (0.71) HPGDTSHRRAB9AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4876 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144801-A1 COMPOSITIONS AND METHODS FOR PREVENTING OR TREATING MUSCLE CONDITIONS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-05-28 US claimed
US-20260137637-A1 ANESTHETIC AGENT MICRO AND NANO PARTICLES, AND METHODS OF MAKING AND USING THE SAME HAAS ERIC (US) 2026-05-21 US claimed
US-12622873-B2 Composition of matter comprising liposomes embedded in a polymeric matrix and methods of using same YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2026-05-12 US claimed
EP-4735042-A1 MERCERIZED DECELLULARIZED PARTICLES FOR SLOW RELEASE APPLICATIONS AND METHODS THEREOF Spiderwort Biotechnologies Inc. (CA) 2026-05-06 EP claimed
US-20260115156-A1 INJECTABLE COMPOSITION INCLUDING HYDROGEL CONTAINING ANESTHETIC AGENT UNIV KOREA RES & BUS FOUND (KR) 2026-04-30 US claimed
US-20260083666-A1 METHOD OF TREATING DISEASE CREWS THOMAS M (US) 2026-03-26 US claimed
EP-4436552-B1 GASTRO-RETENTIVE ORAL DOSAGE UNIT CONTAINING A LOCAL ANAESTHETIC OREXA B V (NL) 2026-02-04 EP claimed
US-12527756-B2 Anesthetic agent micro and nano particles, and methods of making and using the same HAAS ERIC (US) 2026-01-20 US claimed
WO-2025235864-A1 COATED NEEDLE ADMINISTRATION SYSTEMS EVOLUS, INC. (US) 2025-11-13 WO claimed
US-20250319025-A9 COMPOSITIONS COMPRISING MODIFIED PHOSPHOLIPIDS AND USES THEREOF THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-10-16 US claimed
WO-1999055287-A1 TOPICAL ANESTHETIC FORMULATION CASTILLO JAMES (US) 1999-11-04 WO claimed
US-5972326-A Controlled release of pharmaceuticals in the anterior chamber of the eye IOLTECH (FR) 1999-10-26 US claimed
WO-1999022703-A1 IMPROVED PERSONAL CARE FORMULATIONS LURIDENT LTD. (IL) 1999-05-14 WO claimed
WO-1998041171-A1 CONTROLLED RELEASE OF PHARMACEUTICALS IN THE ANTERIOR CHAMBER OF THE EYE GALIN MILES A (US) 1998-09-24 WO claimed
US-5785976-A Solid lipid particles, particles of bioactive agents and methods for the manufacture and use thereof PHARMACIA & UPJOHN AB (SE) 1998-07-28 US claimed
US-5635540-A STABLE MIXTURE OF ETHYLENE OXIDE-PROPYLENE OXIDE COPOLYMER AND WATER AS CARRIER FOR ANTIBIOTICS, FUNGICIDES OR ANESTHETICS, FOR TREATING SKIN DISEASES, BURNS, WOUNDS THE UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 1997-06-03 US claimed
EP-0687172-A1 SOLID LIPID PARTICLES, PARTICLES OF BIOACTIVE AGENTS AND METHODS FOR THE MANUFACTURE AND USE THEREOF Pharmacia & Upjohn Aktiebolag (SE) 1995-12-20 EP claimed
WO-1994020072-A1 SOLID LIPID PARTICLES, PARTICLES OF BIOACTIVE AGENTS AND METHODS FOR THE MANUFACTURE AND USE THEREOF PHARMACIA AB (SE) 1994-09-15 WO claimed
EP-0002426-B1 ANTIPERSPIRANT Playtex-Wallco Aktiebolag (SE) 1981-10-07 EP claimed
EP-0002426-A1 Antiperspirant Playtex-Wallco Aktiebolag (SE) 1979-06-13 EP claimed